
About Course
Medicinal Chemistry.
The main objective of this course is to familiarize students with the fundamental concepts of drug discovery and development. The course is intended for students who have a background in chemistry and interested in the process of drug discovery. The intended outcome is to train students on various aspects of new drug discovery/development, drug screening, target identification, lead discovery, optimization, and the molecular basis of drug design and drug action.
INTENDED AUDIENCE: Third-year undergraduates of B.Sc. Chemistry; M.Sc. Chemistry students and doctoral students
Course Content
Medicinal Chemistry
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Introduction to Medicinal Chemistry Part-I
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Introduction to Medicinal Chemistry Part-II
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Tutorial 01-Acidity, Basicity and Related concepts
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Tutorial 02-Basic Concepts of Thermodynamics and Kinetics
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Tutorial 03- Binding Forces, Protein Structure and Function
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Tutorial 04- Receptors, Binding Interactions, Ion Channels
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Tutorial 05-Nucleic acids, and Basics of Molecular Biology
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Tutorial 06-Enzyme Kinetics, Various Modes of Inhibition etc.
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Tutorial 07-Receptor-Drug Interactions, Stereochemistry, Chirality, Nomenclature
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Tutorial 08-Determination of Drug-Receptor Interactions, Conformation of Cyclic and Acyclic Structur
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Tutorial 09-Nucleic Acids and Related Topics
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Tutorial 10-ADME
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Tutorial 11-Drug administration routes and finding a lead
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Tutorial 12
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Tutorial 13- Optimizing Access-Prodrugs
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Intermolecular Binding Forces
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Protein Structure and Function
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Enzyme Catalysis Part-I
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Enzyme Catalysis Part-II
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Introduction to Receptors
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Receptor Types and Functions
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Enzymes as Drug Targets
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Enzyme Kinetics and Inhibition
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Receptors as Drug Targets Part-I
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Receptors as Drug Targets Part-II
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Pharmacokinetics Part-I
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Pharmacokinetics Part-II
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Finding a Lead Part-I
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Finding a Lead Part-II
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Optimizing Drug-Target Interactions Part-I
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Optimizing Drug-Target Interactions Part-II
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Optimizing Drug-Target Interactions Part-III
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Optimizing Drug-Target Interactions Part-IV
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Endogenous Compounds, Peptidomimetics and Oligonucleotides as Drugs
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Nucleic Acids
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RNA and Protein Synthesis
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Receptor-Drug Interactions.
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Nucleic Acids as Drug Targets Part-I
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Nucleic Acids as Drug Targets Part-II
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Miscellaneous Drug Targets
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Mechanisms in Biological Chemistry Part-I
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Mechanisms in Biological Chemistry Part-II
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Mechanisms in Biological Chemistry Part-III
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Drug Metabolism Part-I
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Drug Metabolism Part-II
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Drug Metabolism Part-III
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Drug Metabolism Part-IV
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Drug Administration Routes Part-I
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Drug Administration Routes Part-II
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Drug Screening
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Optimizing Access to the Target
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Stereochemistry and Conformation
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Prodrugs
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Prodrugs and Drug Alliances
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